Saturday, November 18, 2017

Anabolic Therapies

Anabolic Therapies- Involuntary weight loss is the result of many chronic progressive  diseases, often leading to diminished lean body mass, frailty,  susceptibility to illness, and increased mortality. Various anabolic  agents have been used to combat weight loss with mixed results. Similar  to the frustration experienced by advocates of weight loss in the obese, none of the pharmacological appetite stimulants available at the current  time have been uniformly successful in combating involuntary weight loss in the elderly population. Some of these agents have been U.S. Food and Drug Administration (FDA) approved to combat weight loss, and others are used off-label for this purpose. 
via newspsychology.com

Androgens 


Serum testosterone levels decline with advancing age; however, the  benefits of increasing serum levels by androgen supplementation are controversial. Testosterone has been shown to increase muscle mass  in older men, but adverse effects on the prostate are greater and hematocrit levels are higher than in  younger individuals. Oxandrolone is a chemical derivative of  testosterone that increases muscle mass but has decreased toxicity.  In the elderly, oxandrolone administered daily for 3-month intervals over a year resulted in improved appetite and mental improvement. More recently, the metabolic effects of oxandrolone were thoroughly evaluated in healthy, overweight elderly men.

Highly significant  reductions in abdominal fat were noted, and insulin sensitivity was  improved. Positive effects were most pronounced in men with low testosterone levels, and the benefits were sustained for at least 12  weeks after discontinuation of therapy. Taken together, these  preliminary studies suggest that oxandrolone significantly increases  lean body mass and reduces body fat in healthy elderly men.


Dronabinol (Tetrahydrocannabinol)

Dronabinol, the active ingredient in marijuana, has been used as an  antiemetic and appetite stimulant primarily in cancer and AIDS  patients with mixed results. Little is known about the use of dronabinol in the elderly. Dronabinol, megestrol acetate (MA), and a combination of the two were compared in a randomized study of 469  cancer patients with a mean age of approximately 65 years. MA was superior to dronabinol in terms of appetite (75% vs. 49%) and in the  number of participants who gained more than 10% of their body weight  (11% vs. 3%).
Combination therapy showed no advantage over MA alone.  However, in one intriguing study of 15 Alzheimer's disease patients  hospitalized on a dementia study unit, dronabinol increased body  weight and improved resident behavior. No serious adverse reactions  were noted. Taken together, these studies indicate that dronabinol  is a weak orexigenic (appetitestimulating) agent and is less potent  than MA. There may be a role for its use in treating patients with dementia, but convincing evidence is lacking at the current time.


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